SIMILAR PATTERN OF AMINO ACIDS MAPPED TO '1rjb'

List of Similar Pattern of Amino Acids

Hit pattern: 3D amino acid arrangements similar to known drug binding site

Query pattern: Residues from known binding site for annotated drug that match the hit pattern


(Click on the DrReposER ID to view details on interfaces and similar patterns of amino acids)
(Click on the view link on the last column to view superposed patterns of amino acids)
Filter list by:
DrReposER ID / Desc. Hit
PDBID
Hit
Macromolecule
Res.
Matches
Interface HETATM RMSD Dali
Z-score
Seq.
Identity (%)
View Dock
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1FMO_E_ADNE351_1
(CAMP-DEPENDENT
PROTEIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
GLY A 617
VAL A 624
ALA A 642
VAL A 675
ASN A 816
LEU A 818
None
0.58A 1fmoE-1rjbA:
20.2
1fmoE-1rjbA:
25.06
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1FMO_E_ADNE351_1
(CAMP-DEPENDENT
PROTEIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
VAL A 675
ASN A 816
LEU A 818
ASP A 829
None
0.62A 1fmoE-1rjbA:
20.2
1fmoE-1rjbA:
25.06
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1MUO_A_ADNA1_1
(AURORA-RELATED
KINASE 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 9 LEU A 616
GLY A 617
VAL A 624
ALA A 642
TYR A 693
LEU A 818
None
0.67A 1muoA-1rjbA:
17.2
1muoA-1rjbA:
27.40
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1MXG_A_ACRA443_1
(ALPHA AMYLASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 8 SER A 941
THR A 940
ASN A 938
LYS A 868
None
1.20A 1mxgA-1rjbA:
undetectable
1mxgA-1rjbA:
22.12
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1OPJ_A_STIA3_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
VAL A 675
LEU A 818
None
0.67A 1opjA-1rjbA:
32.5
1opjA-1rjbA:
35.85
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1OPJ_B_STIB4_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
VAL A 675
GLY A 697
ASP A 829
None
0.83A 1opjB-1rjbA:
32.4
1opjB-1rjbA:
35.85
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1SGU_B_MK1B2632_1
(POL POLYPROTEIN)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 8 ALA A 792
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.19A 1sguA-1rjbA:
undetectable
1sguA-1rjbA:
14.24
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1SH9_B_RITB301_1
(POL POLYPROTEIN)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 8 ALA A 792
ILE A 918
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.11A 1sh9A-1rjbA:
undetectable
1sh9A-1rjbA:
14.24
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1T46_A_STIA3_1
(HOMO SAPIENS V-KIT
HARDY-ZUCKERMAN 4
FELINE SARCOMA VIRAL
ONCOGENE HOMOLOG)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
9 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
VAL A 675
GLY A 697
LEU A 818
ASP A 829
None
0.64A 1t46A-1rjbA:
40.4
1t46A-1rjbA:
58.77
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1T46_A_STIA3_2
(HOMO SAPIENS V-KIT
HARDY-ZUCKERMAN 4
FELINE SARCOMA VIRAL
ONCOGENE HOMOLOG)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 7 TYR A 693
CYH A 694
CYH A 807
CYH A 828
None
0.48A 1t46A-1rjbA:
40.4
1t46A-1rjbA:
58.77
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1UWH_A_BAXA1723_1
(B-RAF PROTO-ONCOGENE
SERINE/THREONINE-PRO
TEIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 12 ALA A 642
GLU A 661
CYH A 694
LEU A 802
HIS A 809
None
0.45A 1uwhA-1rjbA:
28.1
1uwhA-1rjbA:
26.59
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1UWH_B_BAXB1723_1
(B-RAF PROTO-ONCOGENE
SERINE/THREONINE-PRO
TEIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 ALA A 642
LYS A 644
GLU A 661
CYH A 694
LEU A 802
HIS A 809
None
0.72A 1uwhB-1rjbA:
27.8
1uwhB-1rjbA:
26.59
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1UWJ_A_BAXA1723_1
(B-RAF PROTO-ONCOGENE
SERINE/THREONINE-PRO
TEIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
CYH A 694
LEU A 802
HIS A 809
None
0.51A 1uwjA-1rjbA:
7.7
1uwjA-1rjbA:
26.59
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1UWJ_B_BAXB1723_1
(B-RAF PROTO-ONCOGENE
SERINE/THREONINE-PRO
TEIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
CYH A 694
LEU A 802
HIS A 809
None
0.51A 1uwjB-1rjbA:
7.7
1uwjB-1rjbA:
26.59
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2EUF_B_LQQB401_1
(CELL DIVISION
PROTEIN KINASE 6)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 VAL A 624
LYS A 644
VAL A 675
PHE A 691
ASP A 698
ASN A 816
LEU A 818
ASP A 829
None
0.91A 2eufB-1rjbA:
22.4
2eufB-1rjbA:
26.60
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2HYY_A_STIA600_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
GLY A 697
LEU A 818
ASP A 829
None
0.76A 2hyyA-1rjbA:
33.5
2hyyA-1rjbA:
37.91
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2HYY_B_STIB600_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
GLY A 697
LEU A 818
ASP A 829
None
0.78A 2hyyB-1rjbA:
33.8
2hyyB-1rjbA:
37.91
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2O4N_A_TPVA300_1
(PROTEASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 12 ALA A 792
ILE A 918
ILE A 921
GLY A 875
PRO A 911
None
0.93A 2o4nA-1rjbA:
undetectable
2o4nA-1rjbA:
14.83
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2O4P_A_TPVA300_1
(PROTEASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 11 ALA A 792
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.09A 2o4pA-1rjbA:
undetectable
2o4pA-1rjbA:
15.12
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2YFX_A_VGHA9000_1
(TYROSINE-PROTEIN
KINASE RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 8 LEU A 616
ALA A 642
GLY A 697
LEU A 818
None
0.58A 2yfxA-1rjbA:
29.3
2yfxA-1rjbA:
36.68
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3C7Q_A_XINA1172_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
9 / 12 LEU A 616
GLY A 617
ALA A 642
LYS A 644
VAL A 675
CYH A 694
GLY A 697
LEU A 818
CYH A 828
None
0.60A 3c7qA-1rjbA:
35.2
3c7qA-1rjbA:
51.96
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3EL4_A_ROCA100_2
(PROTEASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 9 ALA A 792
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.25A 3el4B-1rjbA:
undetectable
3el4B-1rjbA:
14.83
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3EL5_B_1UNB201_1
(PROTEASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 10 ALA A 792
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.17A 3el5A-1rjbA:
undetectable
3el5A-1rjbA:
15.12
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3FUP_B_MI1B1_1
(TYROSINE-PROTEIN
KINASE JAK2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
GLY A 617
VAL A 624
ALA A 642
VAL A 675
TYR A 693
LEU A 818
None
0.53A 3fupB-1rjbA:
27.7
3fupB-1rjbA:
31.94
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3G0E_A_B49A9000_1
(MAST/STEM CELL
GROWTH FACTOR
RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
10 / 11 LEU A 616
VAL A 624
ALA A 642
VAL A 675
TYR A 693
CYH A 694
GLY A 697
LEU A 818
CYH A 828
ALA A 833
None
0.54A 3g0eA-1rjbA:
41.8
3g0eA-1rjbA:
56.77
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3G0F_A_B49A9001_1
(MAST/STEM CELL
GROWTH FACTOR
RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
9 / 11 LEU A 616
VAL A 624
ALA A 642
TYR A 693
CYH A 694
GLY A 697
ASP A 698
LEU A 818
CYH A 828
None
0.55A 3g0fA-1rjbA:
38.5
3g0fA-1rjbA:
56.48
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3G0F_B_B49B9001_1
(MAST/STEM CELL
GROWTH FACTOR
RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 10 LEU A 616
VAL A 624
ALA A 642
TYR A 693
CYH A 694
GLY A 697
LEU A 818
CYH A 828
None
0.48A 3g0fB-1rjbA:
38.8
3g0fB-1rjbA:
56.48
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3G5D_B_1N1B1_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
9 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
VAL A 675
TYR A 693
GLY A 697
LEU A 818
None
0.94A 3g5dB-1rjbA:
29.7
3g5dB-1rjbA:
36.10
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3GVU_A_STIA1001_1
(TYROSINE-PROTEIN
KINASE ABL2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
VAL A 675
LEU A 818
ASP A 829
None
0.82A 3gvuA-1rjbA:
32.1
3gvuA-1rjbA:
38.29
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3IK3_A_0LIA1_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 12 ALA A 642
GLU A 661
HIS A 809
LEU A 818
ASP A 829
None
0.68A 3ik3A-1rjbA:
32.0
3ik3A-1rjbA:
37.57
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3K5V_A_STIA2_1
(TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
GLY A 697
LEU A 818
ASP A 829
None
0.76A 3k5vA-1rjbA:
32.6
3k5vA-1rjbA:
35.85
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3KO0_C_TFPC201_1
(PROTEIN S100-A4)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 9 PHE A 898
GLY A 891
ILE A 876
MET A 855
PHE A 861
None
1.49A 3ko0A-1rjbA:
undetectable
3ko0C-1rjbA:
undetectable
3ko0A-1rjbA:
16.67
3ko0C-1rjbA:
16.67
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3MS9_B_STIB1_1
(TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
GLY A 697
LEU A 818
ASP A 829
None
0.79A 3ms9B-1rjbA:
33.4
3ms9B-1rjbA:
35.85
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3MSS_D_STID1_1
(TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 LEU A 616
ALA A 642
GLU A 661
GLY A 697
LEU A 818
ASP A 829
None
0.76A 3mssD-1rjbA:
33.5
3mssD-1rjbA:
35.85
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3NUO_B_478B478_1
(PROTEASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 9 ALA A 792
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.10A 3nuoA-1rjbA:
undetectable
3nuoA-1rjbA:
14.24
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OCT_A_1N1A663_1
(TYROSINE-PROTEIN
KINASE BTK)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
VAL A 675
TYR A 693
GLY A 697
LEU A 818
None
0.71A 3octA-1rjbA:
29.8
3octA-1rjbA:
36.36
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OCT_A_1N1A663_1
(TYROSINE-PROTEIN
KINASE BTK)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
LYS A 644
MET A 665
VAL A 675
TYR A 693
GLY A 697
LEU A 818
None
1.00A 3octA-1rjbA:
29.8
3octA-1rjbA:
36.36
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OEZ_A_STIA601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 ALA A 642
GLU A 661
VAL A 675
TYR A 693
GLY A 697
LEU A 818
ASP A 829
None
0.71A 3oezA-1rjbA:
30.8
3oezA-1rjbA:
35.82
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OXZ_A_0LIA1_1
(TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 ALA A 642
GLU A 661
VAL A 675
GLY A 697
HIS A 809
ASP A 829
None
0.72A 3oxzA-1rjbA:
31.7
3oxzA-1rjbA:
37.72
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3PYY_B_STIB4_1
(V-ABL ABELSON MURINE
LEUKEMIA VIRAL
ONCOGENE HOMOLOG 1
ISOFORM B VARIANT)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
VAL A 675
LEU A 818
ASP A 829
None
0.82A 3pyyB-1rjbA:
31.1
3pyyB-1rjbA:
35.88
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3QLG_B_1N1B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
VAL A 675
TYR A 693
GLY A 697
LEU A 818
None
0.81A 3qlgB-1rjbA:
29.7
3qlgB-1rjbA:
35.82
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3RGF_A_BAXA465_1
(CYCLIN-DEPENDENT
KINASE 8)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 VAL A 624
ALA A 642
GLU A 661
PHE A 691
TYR A 693
LEU A 802
HIS A 809
None
0.82A 3rgfA-1rjbA:
20.3
3rgfA-1rjbA:
27.33
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3RGF_A_BAXA465_2
(CYCLIN-DEPENDENT
KINASE 8)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 7 LEU A 818
VAL A 675
LEU A 668
ASP A 829
None
0.82A 3rgfA-1rjbA:
20.3
3rgfA-1rjbA:
27.33
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3SXR_A_1N1A1_1
(CYTOPLASMIC
TYROSINE-PROTEIN
KINASE BMX)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
VAL A 675
TYR A 693
GLY A 697
LEU A 818
None
0.52A 3sxrA-1rjbA:
29.1
3sxrA-1rjbA:
36.07
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3SXR_B_1N1B2_1
(CYTOPLASMIC
TYROSINE-PROTEIN
KINASE BMX)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
VAL A 675
TYR A 693
GLY A 697
LEU A 818
None
0.53A 3sxrB-1rjbA:
28.9
3sxrB-1rjbA:
36.07
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3TI1_A_B49A299_1
(CYCLIN-DEPENDENT
KINASE 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 9 ALA A 642
VAL A 675
PHE A 691
ASP A 698
LEU A 818
None
0.71A 3ti1A-1rjbA:
21.3
3ti1A-1rjbA:
26.32
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3U7S_A_017A201_2
(POL POLYPROTEIN)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 9 ALA A 792
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.16A 3u7sB-1rjbA:
undetectable
3u7sB-1rjbA:
15.99
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3WZD_A_LEVA1201_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
GLY A 617
VAL A 624
ALA A 642
GLU A 661
CYH A 694
CYH A 828
None
0.87A 3wzdA-1rjbA:
33.7
3wzdA-1rjbA:
48.27
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3WZD_A_LEVA1201_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
CYH A 694
GLY A 697
CYH A 828
None
0.58A 3wzdA-1rjbA:
33.7
3wzdA-1rjbA:
48.27
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3WZE_A_BAXA1201_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
GLY A 697
LEU A 802
HIS A 809
None
0.60A 3wzeA-1rjbA:
40.1
3wzeA-1rjbA:
48.27
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3WZE_A_BAXA1201_2
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 8 VAL A 675
CYH A 694
LEU A 818
ILE A 827
CYH A 828
ASP A 829
None
0.66A 3wzeA-1rjbA:
40.1
3wzeA-1rjbA:
48.27
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3WZE_A_BAXA1201_2
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 8 VAL A 675
ILE A 827
CYH A 828
ASP A 829
PHE A 830
None
0.83A 3wzeA-1rjbA:
40.1
3wzeA-1rjbA:
48.27
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3ZOS_A_0LIA1000_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
ALA A 642
LYS A 644
GLU A 661
HIS A 809
ARG A 810
LEU A 818
ASP A 829
None
0.87A 3zosA-1rjbA:
32.8
3zosA-1rjbA:
32.11
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3ZOS_A_0LIA1000_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
ALA A 642
LYS A 644
GLU A 661
LEU A 802
HIS A 809
LEU A 818
ASP A 829
None
0.73A 3zosA-1rjbA:
32.8
3zosA-1rjbA:
32.11
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3ZOS_B_0LIB1000_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 ALA A 642
LYS A 644
GLU A 661
LEU A 802
HIS A 809
LEU A 818
ASP A 829
None
0.72A 3zosB-1rjbA:
33.0
3zosB-1rjbA:
32.11
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4AG8_A_AXIA2000_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
9 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
VAL A 675
GLY A 697
LEU A 818
CYH A 828
None
0.53A 4ag8A-1rjbA:
40.2
4ag8A-1rjbA:
48.70
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4AGC_A_AXIA2000_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
GLY A 697
LEU A 818
CYH A 828
None
0.53A 4agcA-1rjbA:
42.2
4agcA-1rjbA:
47.80
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4AGD_A_B49A2000_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 11 LEU A 616
ALA A 642
LYS A 644
VAL A 675
CYH A 694
GLY A 697
LEU A 818
CYH A 828
None
0.65A 4agdA-1rjbA:
41.1
4agdA-1rjbA:
47.80
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4AGD_A_B49A2000_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 11 LYS A 644
VAL A 675
GLY A 697
LEU A 818
CYH A 828
PHE A 830
None
1.26A 4agdA-1rjbA:
41.1
4agdA-1rjbA:
47.80
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4ASD_A_BAXA1500_1
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
GLY A 697
LEU A 802
HIS A 809
None
0.53A 4asdA-1rjbA:
40.6
4asdA-1rjbA:
47.80
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4ASD_A_BAXA1500_2
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 6 VAL A 675
CYH A 694
LEU A 818
ILE A 827
CYH A 828
None
0.55A 4asdA-1rjbA:
40.6
4asdA-1rjbA:
47.80
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4C8B_A_0LIA1000_2
(RECEPTOR-INTERACTING
SERINE/THREONINE-PRO
TEIN KINASE 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 5 VAL A 624
ILE A 674
TYR A 693
ILE A 827
None
0.45A 4c8bA-1rjbA:
25.5
4c8bA-1rjbA:
25.85
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4C8B_B_0LIB1000_1
(RECEPTOR-INTERACTING
SERINE/THREONINE-PRO
TEIN KINASE 2)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 ALA A 642
LYS A 644
GLU A 661
ILE A 674
HIS A 809
LEU A 818
ASP A 829
None
0.85A 4c8bB-1rjbA:
25.3
4c8bB-1rjbA:
25.85
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4CKI_A_ADNA2022_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE RECEPTOR RET)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 11 LEU A 616
GLY A 617
VAL A 624
ALA A 642
TYR A 693
GLY A 697
LEU A 818
None
0.51A 4ckiA-1rjbA:
30.8
4ckiA-1rjbA:
42.77
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4CKI_A_ADNA2022_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE RECEPTOR RET)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 11 LEU A 616
GLY A 831
ALA A 642
TYR A 693
GLY A 697
LEU A 818
None
0.67A 4ckiA-1rjbA:
30.8
4ckiA-1rjbA:
42.77
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4CKJ_A_ADNA2014_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE RECEPTOR RET)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 10 LEU A 616
GLY A 617
GLY A 619
VAL A 624
ALA A 642
TYR A 693
LEU A 818
None
0.55A 4ckjA-1rjbA:
31.5
4ckjA-1rjbA:
43.06
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4IAA_A_RTZA401_1
(SERINE/THREONINE-PRO
TEIN KINASE PIM-1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 11 VAL A 624
ALA A 642
LYS A 644
ASP A 698
LEU A 818
ASP A 829
None
0.83A 4iaaA-1rjbA:
20.4
4iaaA-1rjbA:
24.86
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4L9I_A_8PRA601_1
(RHODOPSIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 7 VAL A 624
ALA A 642
ASP A 698
LEU A 818
None
0.56A 4l9iA-1rjbA:
7.8
4l9iA-1rjbA:
22.27
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4L9I_B_8PRB601_1
(RHODOPSIN KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 8 VAL A 624
ALA A 642
LYS A 644
ASP A 698
LEU A 818
None
0.78A 4l9iB-1rjbA:
20.2
4l9iB-1rjbA:
22.27
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MKC_A_4MKA1503_1
(ALK TYROSINE KINASE
RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLY A 697
ASP A 698
LEU A 818
None
0.55A 4mkcA-1rjbA:
29.5
4mkcA-1rjbA:
36.27
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4O0W_A_ADNA501_1
(AURORA KINASE A)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 6 LEU A 616
GLY A 617
VAL A 624
ALA A 642
LEU A 818
None
0.52A 4o0wA-1rjbA:
22.8
4o0wA-1rjbA:
26.30
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4OGR_E_ADNE401_1
(CYCLIN-DEPENDENT
KINASE 9)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 7 ALA A 642
CYH A 694
ASP A 698
ASN A 816
LEU A 818
ASP A 829
None
0.88A 4ogrE-1rjbA:
21.1
4ogrE-1rjbA:
27.68
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4OGR_E_ADNE401_1
(CYCLIN-DEPENDENT
KINASE 9)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 7 GLY A 617
ALA A 642
CYH A 694
ASP A 698
LEU A 818
None
0.94A 4ogrE-1rjbA:
21.1
4ogrE-1rjbA:
27.68
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4OGR_I_ADNI401_1
(CYCLIN-DEPENDENT
KINASE 9)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 9 GLY A 831
ALA A 642
CYH A 694
ASP A 698
ASN A 816
LEU A 818
None
0.96A 4ogrI-1rjbA:
21.0
4ogrI-1rjbA:
27.68
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4OGR_I_ADNI401_1
(CYCLIN-DEPENDENT
KINASE 9)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 9 GLY A 831
CYH A 694
ASP A 698
ASN A 816
LEU A 818
ASP A 829
None
1.05A 4ogrI-1rjbA:
21.0
4ogrI-1rjbA:
27.68
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4OGR_I_ADNI401_1
(CYCLIN-DEPENDENT
KINASE 9)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 9 VAL A 624
ALA A 642
CYH A 694
ASP A 698
ASN A 816
LEU A 818
None
0.76A 4ogrI-1rjbA:
21.0
4ogrI-1rjbA:
27.68
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4QRC_A_0LIA802_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 4)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 8 LEU A 616
VAL A 624
HIS A 809
LEU A 818
None
0.37A 4qrcA-1rjbA:
33.7
4qrcA-1rjbA:
43.90
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4R7I_A_STIA1001_1
(MACROPHAGE
COLONY-STIMULATING
FACTOR 1 RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 VAL A 624
ALA A 642
LYS A 644
GLU A 661
CYH A 694
CYH A 807
LEU A 818
None
0.61A 4r7iA-1rjbA:
39.9
4r7iA-1rjbA:
55.78
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4R7I_A_STIA1001_1
(MACROPHAGE
COLONY-STIMULATING
FACTOR 1 RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 VAL A 624
ALA A 642
LYS A 644
GLU A 661
CYH A 694
LEU A 818
ASP A 829
None
0.59A 4r7iA-1rjbA:
39.9
4r7iA-1rjbA:
55.78
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4TWP_A_AXIA601_1
(TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLY A 697
ASN A 816
LEU A 818
ASP A 829
None
0.79A 4twpA-1rjbA:
30.5
4twpA-1rjbA:
37.50
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4TYJ_A_0LIA801_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 4)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 6 LEU A 616
VAL A 624
ILE A 674
ILE A 827
None
0.35A 4tyjA-1rjbA:
33.4
4tyjA-1rjbA:
43.60
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4U0I_A_0LIA1001_1
(MAST/STEM CELL
GROWTH FACTOR
RECEPTOR
KIT,MAST/STEM CELL
GROWTH FACTOR
RECEPTOR KIT)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 10 LEU A 616
VAL A 624
GLU A 661
LEU A 668
ILE A 674
VAL A 675
TYR A 693
ILE A 827
None
0.78A 4u0iA-1rjbA:
39.8
4u0iA-1rjbA:
55.52
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4U0I_A_0LIA1001_2
(MAST/STEM CELL
GROWTH FACTOR
RECEPTOR
KIT,MAST/STEM CELL
GROWTH FACTOR
RECEPTOR KIT)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 ALA A 642
LYS A 644
CYH A 694
GLY A 697
HIS A 809
LEU A 818
CYH A 828
ASP A 829
None
0.64A 4u0iA-1rjbA:
39.8
4u0iA-1rjbA:
55.52
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4U5J_A_RXTA601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 11 LEU A 616
VAL A 624
ALA A 642
TYR A 693
GLY A 697
ASN A 816
LEU A 818
ASP A 829
None
0.70A 4u5jA-1rjbA:
30.3
4u5jA-1rjbA:
36.10
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4U5J_B_RXTB601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 9 LEU A 616
VAL A 624
ALA A 642
TYR A 693
GLY A 697
LEU A 818
ASP A 829
None
0.93A 4u5jB-1rjbA:
29.9
4u5jB-1rjbA:
36.10
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4UXQ_A_0LIA1752_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 4)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 LEU A 616
ALA A 642
GLU A 661
LEU A 802
HIS A 809
LEU A 818
None
0.62A 4uxqA-1rjbA:
34.2
4uxqA-1rjbA:
43.90
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V01_A_0LIA1776_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 ALA A 642
GLU A 661
MET A 664
LEU A 802
HIS A 809
ASP A 829
None
0.98A 4v01A-1rjbA:
33.1
4v01A-1rjbA:
45.95
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V01_A_0LIA1776_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 9 LEU A 616
VAL A 624
TYR A 693
CYH A 807
LEU A 818
ILE A 827
None
0.40A 4v01A-1rjbA:
33.1
4v01A-1rjbA:
45.95
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V01_B_0LIB1770_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 ALA A 642
GLU A 661
MET A 664
LEU A 802
HIS A 809
ASP A 829
None
0.93A 4v01B-1rjbA:
33.3
4v01B-1rjbA:
45.95
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V01_B_0LIB1770_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 9 LEU A 616
VAL A 624
LYS A 644
TYR A 693
LEU A 818
ILE A 827
None
0.63A 4v01B-1rjbA:
33.3
4v01B-1rjbA:
45.95
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V04_A_0LIA1772_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
MET A 664
LEU A 802
CYH A 807
None
1.07A 4v04A-1rjbA:
32.8
4v04A-1rjbA:
45.95
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V04_A_0LIA1772_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 VAL A 624
ALA A 642
GLU A 661
MET A 664
LEU A 802
HIS A 809
None
0.90A 4v04A-1rjbA:
32.8
4v04A-1rjbA:
45.95
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V04_B_0LIB1771_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 ALA A 642
GLU A 661
MET A 664
LEU A 802
HIS A 809
ASP A 829
None
1.04A 4v04B-1rjbA:
33.4
4v04B-1rjbA:
45.95
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4ZAU_A_YY3A1101_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 8 LEU A 616
GLY A 617
VAL A 624
ALA A 642
GLY A 697
None
0.66A 4zauA-1rjbA:
29.6
4zauA-1rjbA:
32.38
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5AJQ_A_DB8A800_1
(SERINE/THREONINE-PRO
TEIN KINASE 10)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
ALA A 642
LYS A 644
CYH A 694
GLY A 697
LEU A 818
ASP A 829
None
1.35A 5ajqA-1rjbA:
21.6
5ajqA-1rjbA:
28.33
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5AJQ_A_DB8A800_1
(SERINE/THREONINE-PRO
TEIN KINASE 10)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
GLY A 617
ALA A 642
CYH A 694
GLY A 697
LEU A 818
ASP A 829
None
0.93A 5ajqA-1rjbA:
21.6
5ajqA-1rjbA:
28.33
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5AJQ_B_DB8B800_1
(SERINE/THREONINE-PRO
TEIN KINASE 10)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 10 ALA A 642
CYH A 694
GLY A 697
LEU A 818
ASP A 829
None
0.67A 5ajqB-1rjbA:
21.8
5ajqB-1rjbA:
28.33
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5BVW_A_1N1A1009_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
TYR A 693
GLY A 697
LEU A 818
None
0.78A 5bvwA-1rjbA:
32.3
5bvwA-1rjbA:
31.51
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5HI2_A_BAXA801_1
(SERINE/THREONINE-PRO
TEIN KINASE B-RAF)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 ALA A 642
LYS A 644
GLU A 661
CYH A 694
LEU A 802
HIS A 809
None
0.76A 5hi2A-1rjbA:
27.7
5hi2A-1rjbA:
27.53
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5HI2_A_BAXA801_2
(SERINE/THREONINE-PRO
TEIN KINASE B-RAF)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 8 VAL A 624
ILE A 674
ILE A 827
ASP A 829
None
0.61A 5hi2A-1rjbA:
27.7
5hi2A-1rjbA:
27.53
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5IZJ_F_AZ1F2_1
(CAMP-DEPENDENT
PROTEIN KINASE
CATALYTIC SUBUNIT
ALPHA
47P-AZ1-DAR-DAR-DAR)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 7 GLY A 617
GLY A 619
GLY A 622
VAL A 624
None
0.30A 5izjB-1rjbA:
20.8
5izjB-1rjbA:
24.69
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5KR0_A_478A101_1
(PROTEASE E35D-APV)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 9 ALA A 792
ILE A 921
GLY A 875
ILE A 876
PRO A 911
None
1.03A 5kr0A-1rjbA:
undetectable
5kr0A-1rjbA:
14.24
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5L2I_A_LQQA900_1
(CYCLIN-DEPENDENT
KINASE 6)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 GLY A 617
VAL A 624
ALA A 642
VAL A 675
PHE A 691
ASP A 698
LEU A 818
None
0.60A 5l2iA-1rjbA:
6.6
5l2iA-1rjbA:
25.86
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5L2T_A_6ZZA900_1
(CYCLIN-DEPENDENT
KINASE 6)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 GLY A 617
VAL A 624
ALA A 642
VAL A 675
PHE A 691
ASP A 698
LEU A 818
None
0.86A 5l2tA-1rjbA:
6.6
5l2tA-1rjbA:
25.86
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5LVN_A_ADNA402_1
(3-PHOSPHOINOSITIDE-D
EPENDENT PROTEIN
KINASE 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 11 LEU A 616
GLY A 617
VAL A 624
ALA A 642
VAL A 675
TYR A 693
LEU A 818
None
0.47A 5lvnA-1rjbA:
21.9
5lvnA-1rjbA:
25.88
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5MAF_A_XINA403_1
(MATERNAL EMBRYONIC
LEUCINE ZIPPER
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 GLY A 617
VAL A 624
ALA A 642
LYS A 644
GLU A 661
TYR A 693
GLY A 697
None
0.71A 5mafA-1rjbA:
22.1
5mafA-1rjbA:
12.42
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5OWR_A_1N1A401_1
(SERINE/THREONINE-PRO
TEIN KINASE 10)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 8 ALA A 642
GLU A 661
CYH A 694
LEU A 818
None
0.48A 5owrA-1rjbA:
19.6
5owrA-1rjbA:
26.46
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5TE0_A_XINA401_2
(AP2-ASSOCIATED
PROTEIN KINASE 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 5 LEU A 616
VAL A 624
CYH A 694
CYH A 828
None
0.58A 5te0A-1rjbA:
21.8
5te0A-1rjbA:
23.04
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5VC3_A_DB8A601_1
(WEE1-LIKE PROTEIN
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 GLY A 617
ALA A 642
GLU A 661
TYR A 693
CYH A 694
GLY A 697
ASP A 829
None
0.79A 5vc3A-1rjbA:
21.9
5vc3A-1rjbA:
24.44
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5VCV_A_1N1A404_1
(MEMBRANE-ASSOCIATED
TYROSINE- AND
THREONINE-SPECIFIC
CDC2-INHIBITORY
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 LEU A 616
ALA A 642
GLU A 661
VAL A 675
LEU A 689
GLY A 697
None
1.09A 5vcvA-1rjbA:
21.9
5vcvA-1rjbA:
25.34
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5VCV_A_1N1A404_1
(MEMBRANE-ASSOCIATED
TYROSINE- AND
THREONINE-SPECIFIC
CDC2-INHIBITORY
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 LEU A 616
ALA A 642
LYS A 644
GLU A 661
LEU A 689
GLY A 697
None
1.39A 5vcvA-1rjbA:
21.9
5vcvA-1rjbA:
25.34
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5VCY_A_DB8A401_1
(MEMBRANE-ASSOCIATED
TYROSINE- AND
THREONINE-SPECIFIC
CDC2-INHIBITORY
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
LEU A 689
CYH A 694
None
0.70A 5vcyA-1rjbA:
21.6
5vcyA-1rjbA:
25.34
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5VCY_A_DB8A401_1
(MEMBRANE-ASSOCIATED
TYROSINE- AND
THREONINE-SPECIFIC
CDC2-INHIBITORY
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
6 / 12 LEU A 616
VAL A 624
ALA A 642
LYS A 644
GLU A 661
LEU A 689
None
0.93A 5vcyA-1rjbA:
21.6
5vcyA-1rjbA:
25.34
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5W5V_A_ANWA701_0
(SERINE/THREONINE-PRO
TEIN KINASE TBK1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 9 LEU A 616
ALA A 642
VAL A 675
CYH A 694
GLY A 697
None
0.49A 5w5vA-1rjbA:
13.4
5w5vA-1rjbA:
20.97
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5XV7_A_EMHA705_1
(SERINE-ARGININE (SR)
PROTEIN KINASE 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
5 / 12 LEU A 616
GLY A 617
VAL A 624
ALA A 642
PHE A 691
None
0.45A 5xv7A-1rjbA:
19.8
5xv7A-1rjbA:
12.57
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5Y7Z_A_IREA401_0
(CYCLIN-G-ASSOCIATED
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
CYH A 694
GLY A 697
LEU A 818
None
0.57A 5y7zA-1rjbA:
21.1
5y7zA-1rjbA:
12.82
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5Y7Z_A_IREA401_0
(CYCLIN-G-ASSOCIATED
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
CYH A 694
GLY A 697
LEU A 818
None
0.57A 5y7zA-1rjbA:
21.1
5y7zA-1rjbA:
24.93
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5Y7Z_B_IREB401_0
(CYCLIN-G-ASSOCIATED
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
ALA A 642
GLU A 661
CYH A 694
GLY A 697
LEU A 818
CYH A 828
ASP A 829
None
0.87A 5y7zB-1rjbA:
21.2
5y7zB-1rjbA:
12.82
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5Y80_A_IREA401_0
(CYCLIN-G-ASSOCIATED
KINASE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
8 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
CYH A 694
GLY A 697
LEU A 818
ASP A 829
None
0.75A 5y80A-1rjbA:
20.8
5y80A-1rjbA:
12.82
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5Y9M_A_NIOA401_1
(CASEIN KINASE II
SUBUNIT ALPHA')
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
4 / 8 LEU A 616
VAL A 624
LYS A 644
PHE A 691
None
0.71A 5y9mA-1rjbA:
20.1
5y9mA-1rjbA:
16.36
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5ZV2_A_LEVA801_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
GLY A 617
VAL A 624
ALA A 642
GLU A 661
TYR A 693
GLY A 697
None
0.88A 5zv2A-1rjbA:
32.7
5zv2A-1rjbA:
15.06
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5ZV2_B_LEVB801_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
GLY A 617
VAL A 624
ALA A 642
LYS A 644
GLU A 661
GLY A 697
None
1.01A 5zv2B-1rjbA:
32.3
5zv2B-1rjbA:
15.06
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6ECE_C_DVAC3010_0
(VLM2
DODECADEPSIPEPTIDE)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
3 / 3 ALA A 856
PHE A 928
GLN A 903
None
0.82A 6eceA-1rjbA:
undetectable
6eceA-1rjbA:
21.25
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6HD6_B_STIB601_0
(TYROSINE-PROTEIN
KINASE ABL1)
1rjb FL CYTOKINE RECEPTOR
(Homo
sapiens)
7 / 12 LEU A 616
VAL A 624
ALA A 642
GLU A 661
VAL A 675
LEU A 818
ASP A 829
None
0.85A 6hd6B-1rjbA:
32.3
6hd6B-1rjbA:
13.17