SIMILAR PATTERN OF AMINO ACIDS MAPPED TO '3kex'

List of Similar Pattern of Amino Acids

Hit pattern: 3D amino acid arrangements similar to known drug binding site

Query pattern: Residues from known binding site for annotated drug that match the hit pattern


(Click on the DrReposER ID to view details on interfaces and similar patterns of amino acids)
(Click on the view link on the last column to view superposed patterns of amino acids)
Filter list by:
DrReposER ID / Desc. Hit
PDBID
Hit
Macromolecule
Res.
Matches
Interface HETATM RMSD Dali
Z-score
Seq.
Identity (%)
View Dock
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1M17_A_AQ4A999_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
LYS A 723
LEU A 766
THR A 768
GLY A 774
LEU A 822
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.84A 1m17A-3kexA:
32.0
1m17A-3kexA:
54.05
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XKK_A_FMMA91_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 THR A 768
GLY A 774
LEU A 777
ASP A 778
ARG A 781
LEU A 822
ASP A 833
PHE A 834
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
None
None
None
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
None
0.56A 1xkkA-3kexA:
36.0
1xkkA-3kexA:
51.14
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XKK_A_FMMA91_2
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 9 LEU A 696
VAL A 704
LYS A 723
LEU A 755
LEU A 766
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
None
0.40A 1xkkA-3kexA:
36.0
1xkkA-3kexA:
51.14
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2GQG_B_1N1B502_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.47A 2gqgB-3kexA:
28.2
2gqgB-3kexA:
35.47
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ITO_A_IREA2020_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
LYS A 723
LEU A 766
THR A 768
GLY A 774
ASP A 778
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
None
ANP  A   1 (-4.7A)
0.57A 2itoA-3kexA:
31.7
2itoA-3kexA:
54.74
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ITY_A_IREA2020_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
GLY A 697
VAL A 704
LYS A 723
LEU A 766
THR A 768
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.7A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.71A 2ityA-3kexA:
31.8
2ityA-3kexA:
55.05
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ITZ_A_IREA2021_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
LYS A 723
THR A 768
GLY A 774
ASP A 778
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
None
ANP  A   1 (-4.7A)
0.68A 2itzA-3kexA:
31.8
2itzA-3kexA:
55.05
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ZVA_A_1N1A513_1
(TYROSINE-PROTEIN
KINASE LYN)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
LYS A 723
VAL A 753
THR A 768
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.69A 2zvaA-3kexA:
27.9
2zvaA-3kexA:
32.22
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3BBT_B_FMMB91_1
(RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-4)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 VAL A 704
LEU A 755
THR A 768
GLY A 774
LEU A 822
ASP A 833
PHE A 834
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
None
0.53A 3bbtB-3kexA:
32.4
3bbtB-3kexA:
58.41
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3BBT_D_FMMD91_1
(RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-4)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 VAL A 704
LYS A 723
LEU A 766
THR A 768
GLY A 774
LEU A 822
ASP A 833
PHE A 834
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
None
0.61A 3bbtD-3kexA:
36.0
3bbtD-3kexA:
58.41
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3CE6_D_ADND500_2
(ADENOSYLHOMOCYSTEINA
SE)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
4 / 5 LEU A 773
GLN A 828
HIS A 783
LEU A 787
None
0.90A 3ce6D-3kexA:
undetectable
3ce6D-3kexA:
20.16
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3CS9_B_NILB600_2
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 9 LEU A 696
VAL A 704
VAL A 753
LEU A 822
VAL A 831
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 (-4.7A)
None
0.79A 3cs9B-3kexA:
25.3
3cs9B-3kexA:
35.59
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3CS9_C_NILC600_2
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 9 LEU A 696
VAL A 704
LYS A 723
VAL A 753
VAL A 831
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
None
1.10A 3cs9C-3kexA:
24.4
3cs9C-3kexA:
35.59
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3EYG_A_MI1A1_1
(TYROSINE-PROTEIN
KINASE)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
9 / 12 LEU A 696
GLY A 699
GLY A 702
VAL A 704
LYS A 723
SER A 775
ASN A 820
LEU A 822
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 (-2.8A)
None
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 2.6A)
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.87A 3eygA-3kexA:
28.1
3eygA-3kexA:
30.33
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3G0F_A_B49A9001_1
(MAST/STEM CELL
GROWTH FACTOR
RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 11 LEU A 696
VAL A 704
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.72A 3g0fA-3kexA:
26.3
3g0fA-3kexA:
28.31
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3G0F_B_B49B9001_1
(MAST/STEM CELL
GROWTH FACTOR
RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 10 LEU A 696
VAL A 704
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.63A 3g0fB-3kexA:
26.7
3g0fB-3kexA:
28.31
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3G5D_A_1N1A1_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.55A 3g5dA-3kexA:
28.5
3g5dA-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3G5D_B_1N1B1_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
9 / 12 LEU A 696
VAL A 704
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.68A 3g5dB-3kexA:
28.4
3g5dB-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3GVU_A_STIA1001_1
(TYROSINE-PROTEIN
KINASE ABL2)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.7A)
None
0.64A 3gvuA-3kexA:
24.6
3gvuA-3kexA:
35.92
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3K54_A_1N1A1_1
(TYROSINE-PROTEIN
KINASE BTK)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.50A 3k54A-3kexA:
27.7
3k54A-3kexA:
28.19
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3MS9_B_STIB1_1
(TYROSINE-PROTEIN
KINASE ABL1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 12 LEU A 696
VAL A 704
THR A 768
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.64A 3ms9B-3kexA:
27.3
3ms9B-3kexA:
33.84
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3OCT_A_1N1A663_1
(TYROSINE-PROTEIN
KINASE BTK)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
VAL A 704
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.54A 3octA-3kexA:
27.2
3octA-3kexA:
28.66
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OEZ_A_STIA601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 VAL A 704
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.73A 3oezA-3kexA:
27.8
3oezA-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3PYY_B_STIB4_1
(V-ABL ABELSON MURINE
LEUKEMIA VIRAL
ONCOGENE HOMOLOG 1
ISOFORM B VARIANT)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.7A)
None
0.72A 3pyyB-3kexA:
28.0
3pyyB-3kexA:
32.73
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3QLG_A_1N1A601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.64A 3qlgA-3kexA:
28.2
3qlgA-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3QLG_A_1N1A601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 VAL A 704
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.81A 3qlgA-3kexA:
28.2
3qlgA-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3QLG_B_1N1B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
9 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
MG  A1001 ( 3.1A)
0.68A 3qlgB-3kexA:
28.5
3qlgB-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3SXR_A_1N1A1_1
(CYTOPLASMIC
TYROSINE-PROTEIN
KINASE BMX)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.48A 3sxrA-3kexA:
27.6
3sxrA-3kexA:
31.58
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3SXR_B_1N1B2_1
(CYTOPLASMIC
TYROSINE-PROTEIN
KINASE BMX)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.46A 3sxrB-3kexA:
27.2
3sxrB-3kexA:
31.58
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3UG2_A_IREA1_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
LYS A 723
LEU A 766
GLY A 774
ASP A 778
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.9A)
None
ANP  A   1 (-4.7A)
0.67A 3ug2A-3kexA:
31.7
3ug2A-3kexA:
53.59
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3WZD_A_LEVA1201_2
(VASCULAR ENDOTHELIAL
GROWTH FACTOR
RECEPTOR 2)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
4 / 5 ILE A 744
VAL A 753
LEU A 822
ASP A 833
None
None
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.58A 3wzdA-3kexA:
27.3
3wzdA-3kexA:
28.57
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4CKI_A_ADNA2022_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE RECEPTOR RET)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 11 LEU A 696
GLY A 697
VAL A 704
TYR A 770
GLY A 774
SER A 775
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.7A)
ANP  A   1 (-3.9A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
None
ANP  A   1 (-4.7A)
0.75A 4ckiA-3kexA:
28.9
4ckiA-3kexA:
28.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4HJO_A_AQ4A1001_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
LYS A 723
THR A 768
GLY A 774
LEU A 822
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.53A 4hjoA-3kexA:
36.0
4hjoA-3kexA:
53.12
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4I22_A_IREA9001_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
9 / 12 LEU A 696
GLY A 697
VAL A 704
LYS A 723
LEU A 766
GLY A 774
ASP A 778
LEU A 822
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 (-3.7A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.9A)
None
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.75A 4i22A-3kexA:
35.5
4i22A-3kexA:
54.10
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4IFG_A_1E8A601_1
(CALMODULIN-DOMAIN
PROTEIN KINASE 1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 GLY A 697
VAL A 704
LYS A 723
LEU A 755
LEU A 766
GLY A 774
LEU A 822
ANP  A   1 (-3.7A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
None
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.73A 4ifgA-3kexA:
24.3
4ifgA-3kexA:
21.14
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4LMN_A_EUIA503_1
(DUAL SPECIFICITY
MITOGEN-ACTIVATED
PROTEIN KINASE
KINASE 1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 12 LYS A 723
ASN A 820
ASP A 833
PHE A 834
LEU A 839
ANP  A   1 (-3.4A)
ANP  A   1 ( 2.6A)
MG  A1001 ( 3.1A)
None
None
0.83A 4lmnA-3kexA:
24.0
4lmnA-3kexA:
24.11
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4MJ8_A_SPMA202_1
(SPERMIDINE
N1-ACETYLTRANSFERASE)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 8 GLU A 687
ILE A 722
GLN A 765
ILE A 725
LEU A 758
None
1.47A 4mj8A-3kexA:
undetectable
4mj8A-3kexA:
19.51
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXO_A_DB8A601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
0.67A 4mxoA-3kexA:
28.1
4mxoA-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXO_B_DB8B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
VAL A 704
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.66A 4mxoB-3kexA:
27.7
4mxoB-3kexA:
33.03
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXX_A_DB8A601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.58A 4mxxA-3kexA:
28.0
4mxxA-3kexA:
32.73
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXX_B_DB8B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
VAL A 704
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.55A 4mxxB-3kexA:
27.7
4mxxB-3kexA:
32.73
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXY_B_DB8B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
VAL A 753
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.67A 4mxyB-3kexA:
26.5
4mxyB-3kexA:
32.73
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXZ_B_DB8B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
VAL A 753
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
None
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.67A 4mxzB-3kexA:
26.5
4mxzB-3kexA:
32.73
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4OTW_A_DB8A1101_1
(RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
12 / 12 LEU A 696
VAL A 704
CYH A 721
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ASP A 833
VAL A 836
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.5A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
MG  A1001 ( 3.1A)
None
0.49A 4otwA-3kexA:
42.2
4otwA-3kexA:
99.69
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4RZV_B_032B801_1
(SERINE/THREONINE-PRO
TEIN KINASE B-RAF)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 12 VAL A 704
LYS A 723
THR A 768
SER A 775
PHE A 834
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
ANP  A   1 ( 4.8A)
None
None
0.85A 4rzvB-3kexA:
27.5
4rzvB-3kexA:
29.18
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4WKQ_A_IREA1101_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
LYS A 723
LEU A 766
THR A 768
GLY A 774
ASP A 778
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
None
ANP  A   1 (-4.7A)
0.61A 4wkqA-3kexA:
32.4
4wkqA-3kexA:
54.85
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XEY_A_1N1A601_1
(TYROSINE-PROTEIN
KINASE ABL1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
VAL A 704
LYS A 723
VAL A 753
THR A 768
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.55A 4xeyA-3kexA:
27.2
4xeyA-3kexA:
28.18
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XEY_B_1N1B601_1
(TYROSINE-PROTEIN
KINASE ABL1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
LYS A 723
THR A 768
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.55A 4xeyB-3kexA:
21.4
4xeyB-3kexA:
28.18
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XEY_B_1N1B601_1
(TYROSINE-PROTEIN
KINASE ABL1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
VAL A 704
LYS A 723
VAL A 753
THR A 768
GLY A 774
LEU A 822
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
0.38A 4xeyB-3kexA:
21.4
4xeyB-3kexA:
28.18
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4XLI_A_1N1A601_1
(NON-SPECIFIC
PROTEIN-TYROSINE
KINASE)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.60A 4xliA-3kexA:
24.8
4xliA-3kexA:
36.55
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4XLI_B_1N1B600_1
(NON-SPECIFIC
PROTEIN-TYROSINE
KINASE)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
LYS A 723
VAL A 753
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.66A 4xliB-3kexA:
28.7
4xliB-3kexA:
36.55
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5BVW_A_1N1A1009_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
8 / 12 LEU A 696
VAL A 704
LYS A 723
THR A 768
TYR A 770
GLY A 774
LEU A 822
ALA A 832
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
None
0.67A 5bvwA-3kexA:
27.0
5bvwA-3kexA:
30.89
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5D4N_C_ACTC201_0
(NITROGEN REGULATORY
PROTEIN P-II)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
4 / 5 VAL A 921
VAL A 882
GLY A 879
PHE A 946
None
1.08A 5d4nA-3kexA:
undetectable
5d4nC-3kexA:
undetectable
5d4nA-3kexA:
18.75
5d4nC-3kexA:
18.75
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5H2U_B_1N1B501_1
(PROTEIN-TYROSINE
KINASE 6)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 12 LEU A 696
VAL A 704
THR A 768
GLY A 774
LEU A 822
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 (-3.9A)
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.73A 5h2uB-3kexA:
33.4
5h2uB-3kexA:
30.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5H2U_C_1N1C501_1
(PROTEIN-TYROSINE
KINASE 6)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 12 LEU A 696
THR A 768
GLY A 774
LEU A 822
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 ( 4.8A)
ANP  A   1 ( 4.9A)
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.59A 5h2uC-3kexA:
33.2
5h2uC-3kexA:
30.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5HES_A_032A401_1
(MITOGEN-ACTIVATED
PROTEIN KINASE
KINASE KINASE MLT)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 12 VAL A 704
THR A 768
TYR A 770
ASP A 778
PHE A 834
ANP  A   1 (-3.9A)
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
None
None
0.70A 5hesA-3kexA:
27.1
5hesA-3kexA:
30.92
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5HES_B_032B401_1
(MITOGEN-ACTIVATED
PROTEIN KINASE
KINASE KINASE MLT)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 12 VAL A 704
LYS A 723
THR A 768
TYR A 770
ASP A 778
PHE A 834
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
ANP  A   1 ( 4.8A)
ANP  A   1 (-4.3A)
None
None
0.78A 5hesB-3kexA:
26.6
5hesB-3kexA:
30.92
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5IZJ_F_AZ1F2_1
(CAMP-DEPENDENT
PROTEIN KINASE
CATALYTIC SUBUNIT
ALPHA
47P-AZ1-DAR-DAR-DAR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
5 / 7 GLY A 697
GLY A 699
PHE A 701
GLY A 702
VAL A 704
ANP  A   1 (-3.7A)
ANP  A   1 (-2.8A)
None
None
ANP  A   1 (-3.9A)
0.56A 5izjB-3kexA:
19.4
5izjB-3kexA:
25.13
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5YU9_A_1E8A1101_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 LEU A 696
GLY A 697
VAL A 704
LYS A 723
LEU A 766
LEU A 822
ASP A 833
ANP  A   1 (-4.4A)
ANP  A   1 (-3.7A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.60A 5yu9A-3kexA:
35.4
5yu9A-3kexA:
15.79
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5YU9_B_1E8B1101_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
7 / 12 GLY A 697
VAL A 704
LYS A 723
LEU A 766
ASP A 778
LEU A 822
ASP A 833
ANP  A   1 (-3.7A)
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
None
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.83A 5yu9B-3kexA:
35.1
5yu9B-3kexA:
15.79
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5YU9_C_1E8C1101_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 12 VAL A 704
LYS A 723
LEU A 766
GLY A 774
ASP A 778
ASP A 833
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
None
ANP  A   1 ( 4.9A)
None
MG  A1001 ( 3.1A)
0.70A 5yu9C-3kexA:
30.1
5yu9C-3kexA:
15.79
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5YU9_D_1E8D1101_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3kex RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3

(Homo
sapiens)
6 / 12 VAL A 704
LYS A 723
GLY A 774
ASP A 778
LEU A 822
ASP A 833
ANP  A   1 (-3.9A)
ANP  A   1 (-3.4A)
ANP  A   1 ( 4.9A)
None
ANP  A   1 (-4.7A)
MG  A1001 ( 3.1A)
0.81A 5yu9D-3kexA:
30.4
5yu9D-3kexA:
15.79