SIMILAR PATTERN OF AMINO ACIDS MAPPED TO '3s95'

List of Similar Pattern of Amino Acids

Hit pattern: 3D amino acid arrangements similar to known drug binding site

Query pattern: Residues from known binding site for annotated drug that match the hit pattern


(Click on the DrReposER ID to view details on interfaces and similar patterns of amino acids)
(Click on the view link on the last column to view superposed patterns of amino acids)
Filter list by:
DrReposER ID / Desc. Hit
PDBID
Hit
Macromolecule
Res.
Matches
Interface HETATM RMSD Dali
Z-score
Seq.
Identity (%)
View Dock
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1HWI_C_115C4_1
(HMG-COA REDUCTASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
4 / 7 ARG A 608
VAL A 438
SER A 439
ASN A 473
None
1.21A 1hwiC-3s95A:
undetectable
1hwiC-3s95A:
22.12
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1HWI_D_115D3_2
(HMG-COA REDUCTASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
4 / 7 ARG A 608
VAL A 438
SER A 439
ASN A 473
None
1.21A 1hwiD-3s95A:
undetectable
1hwiD-3s95A:
22.12
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1IEP_A_STIA201_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
GLU A 384
MET A 388
THR A 413
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
1.06A 1iepA-3s95A:
24.1
1iepA-3s95A:
31.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1OPJ_B_STIB4_2
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
4 / 6 LEU A 345
LYS A 368
VAL A 387
ARG A 459
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
None
None
1.00A 1opjB-3s95A:
23.6
1opjB-3s95A:
31.37
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1QOM_A_H4BA902_1
(NITRIC OXIDE
SYNTHASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 ARG A 422
ILE A 537
TRP A 515
TRS  A 640 (-3.9A)
None
None
1.12A 1qomA-3s95A:
undetectable
1qomA-3s95A:
22.00
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1QW6_A_H4BA901_1
(NITRIC-OXIDE
SYNTHASE, BRAIN)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 ARG A 555
VAL A 538
TRP A 515
GOL  A   4 ( 3.9A)
None
None
1.24A 1qw6A-3s95A:
undetectable
1qw6A-3s95A:
21.14
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1QWC_A_H4BA901_1
(NITRIC-OXIDE
SYNTHASE, BRAIN)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 ARG A 555
VAL A 538
TRP A 515
GOL  A   4 ( 3.9A)
None
None
1.22A 1qwcA-3s95A:
undetectable
1qwcA-3s95A:
21.14
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1UWH_A_BAXA1723_1
(B-RAF PROTO-ONCOGENE
SERINE/THREONINE-PRO
TEIN KINASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 12 GLU A 384
LEU A 397
THR A 413
LEU A 451
HIS A 458
STU  A   1 (-3.7A)
STU  A   1 (-4.6A)
STU  A   1 (-3.9A)
None
None
0.62A 1uwhA-3s95A:
26.3
1uwhA-3s95A:
29.57
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1UWH_B_BAXB1723_1
(B-RAF PROTO-ONCOGENE
SERINE/THREONINE-PRO
TEIN KINASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 12 LYS A 368
GLU A 384
LEU A 397
THR A 413
LEU A 451
HIS A 458
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-4.6A)
STU  A   1 (-3.9A)
None
None
0.70A 1uwhB-3s95A:
26.1
1uwhB-3s95A:
29.57
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1VAG_A_H4BA901_1
(NITRIC-OXIDE
SYNTHASE, BRAIN)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 ARG A 555
VAL A 538
TRP A 515
GOL  A   4 ( 3.9A)
None
None
1.21A 1vagA-3s95A:
undetectable
1vagA-3s95A:
21.14
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2GQG_A_1N1A501_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
LYS A 368
GLU A 384
THR A 413
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.81A 2gqgA-3s95A:
20.2
2gqgA-3s95A:
31.06
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2GQG_A_1N1A501_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
GLU A 384
MET A 388
THR A 413
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.70A 2gqgA-3s95A:
20.2
2gqgA-3s95A:
31.06
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2HYY_C_STIC600_2
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
4 / 6 LEU A 345
LYS A 368
VAL A 387
MET A 388
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
None
None
0.88A 2hyyC-3s95A:
24.5
2hyyC-3s95A:
30.75
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2ITO_A_IREA2020_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
LYS A 368
GLU A 384
MET A 388
THR A 413
GLY A 419
LEU A 467
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.99A 2itoA-3s95A:
27.1
2itoA-3s95A:
27.79
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2OIQ_A_STIA1001_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.96A 2oiqA-3s95A:
24.8
2oiqA-3s95A:
35.14
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2WGJ_A_VGHA2346_1
(HEPATOCYTE GROWTH
FACTOR RECEPTOR)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 12 GLY A 346
LEU A 397
TYR A 415
GLY A 419
ALA A 477
ASP A 478
STU  A   1 (-3.4A)
STU  A   1 (-4.6A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 ( 4.1A)
STU  A   1 ( 4.2A)
0.75A 2wgjA-3s95A:
24.4
2wgjA-3s95A:
30.40
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2Y6O_A_1N1A1892_1
(EPHRIN TYPE-A
RECEPTOR 4)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.84A 2y6oA-3s95A:
20.1
2y6oA-3s95A:
29.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2ZBZ_A_VDXA501_1
(CYTOCHROME P450-SU1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 11 THR A 413
VAL A 387
MET A 454
ILE A 456
ALA A 477
STU  A   1 (-3.9A)
None
None
None
STU  A   1 ( 4.1A)
1.11A 2zbzA-3s95A:
undetectable
2zbzA-3s95A:
21.82
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ZVA_A_1N1A513_1
(TYROSINE-PROTEIN
KINASE LYN)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
LYS A 368
GLU A 384
THR A 413
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.78A 2zvaA-3s95A:
27.5
2zvaA-3s95A:
30.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ZVA_A_1N1A513_1
(TYROSINE-PROTEIN
KINASE LYN)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
GLU A 384
MET A 388
THR A 413
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.69A 2zvaA-3s95A:
27.5
2zvaA-3s95A:
30.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3G5D_B_1N1B1_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.77A 3g5dB-3s95A:
26.5
3g5dB-3s95A:
35.14
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3MS9_B_STIB1_1
(TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
GLU A 384
MET A 388
THR A 413
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
1.07A 3ms9B-3s95A:
23.6
3ms9B-3s95A:
31.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3MSS_A_STIA1_1
(TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 12 LEU A 345
GLU A 384
MET A 388
THR A 413
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
1.13A 3mssA-3s95A:
24.0
3mssA-3s95A:
31.37
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3MSS_D_STID1_1
(TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
GLU A 384
MET A 388
THR A 413
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
1.09A 3mssD-3s95A:
23.8
3mssD-3s95A:
31.37
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3NW2_A_H4BA902_1
(NITRIC OXIDE
SYNTHASE, INDUCIBLE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 ARG A 422
ILE A 537
TRP A 515
TRS  A 640 (-3.9A)
None
None
1.13A 3nw2A-3s95A:
undetectable
3nw2A-3s95A:
21.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3NW2_B_H4BB902_1
(NITRIC OXIDE
SYNTHASE, INDUCIBLE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 ARG A 422
ILE A 537
TRP A 515
TRS  A 640 (-3.9A)
None
None
1.10A 3nw2B-3s95A:
undetectable
3nw2B-3s95A:
21.72
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OEZ_B_STIB601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
VAL A 387
MET A 388
THR A 413
TYR A 415
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
None
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.89A 3oezB-3s95A:
24.9
3oezB-3s95A:
34.83
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OXZ_A_0LIA1_2
(TYROSINE-PROTEIN
KINASE ABL1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 9 LEU A 345
LYS A 368
VAL A 387
ARG A 459
LEU A 467
VAL A 476
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
None
None
STU  A   1 (-4.6A)
None
1.04A 3oxzA-3s95A:
25.0
3oxzA-3s95A:
30.65
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3QLG_A_1N1A601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
9 / 12 LEU A 345
LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.86A 3qlgA-3s95A:
25.8
3qlgA-3s95A:
34.83
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3QLG_B_1N1B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LEU A 345
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.76A 3qlgB-3s95A:
26.4
3qlgB-3s95A:
34.83
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3SXR_A_1N1A1_1
(CYTOPLASMIC
TYROSINE-PROTEIN
KINASE BMX)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
MET A 388
THR A 413
TYR A 415
ILE A 416
GLY A 419
LEU A 467
STU  A   1 (-3.8A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-4.3A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.61A 3sxrA-3s95A:
25.6
3sxrA-3s95A:
30.13
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3SXR_B_1N1B2_1
(CYTOPLASMIC
TYROSINE-PROTEIN
KINASE BMX)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
MET A 388
THR A 413
TYR A 415
ILE A 416
GLY A 419
LEU A 467
STU  A   1 (-3.8A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-4.3A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.61A 3sxrB-3s95A:
25.2
3sxrB-3s95A:
30.13
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3ZOS_A_0LIA1000_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
9 / 12 LEU A 345
LYS A 368
GLU A 384
THR A 413
LEU A 451
HIS A 458
ARG A 459
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-3.9A)
None
None
None
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.94A 3zosA-3s95A:
24.1
3zosA-3s95A:
29.13
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3ZOS_B_0LIB1000_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LYS A 368
GLU A 384
THR A 413
LEU A 451
HIS A 458
ARG A 459
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-3.9A)
None
None
None
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
1.01A 3zosB-3s95A:
24.2
3zosB-3s95A:
29.13
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4C8B_A_0LIA1000_1
(RECEPTOR-INTERACTING
SERINE/THREONINE-PRO
TEIN KINASE 2)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
GLU A 384
LEU A 397
THR A 413
HIS A 458
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-4.6A)
STU  A   1 (-3.9A)
None
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.75A 4c8bA-3s95A:
25.4
4c8bA-3s95A:
23.81
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4C8B_B_0LIB1000_1
(RECEPTOR-INTERACTING
SERINE/THREONINE-PRO
TEIN KINASE 2)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
GLU A 384
LEU A 397
THR A 413
HIS A 458
LEU A 467
ALA A 477
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-4.6A)
STU  A   1 (-3.9A)
None
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.79A 4c8bB-3s95A:
25.2
4c8bB-3s95A:
23.81
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4MJ8_A_SPMA202_1
(SPERMIDINE
N1-ACETYLTRANSFERASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
4 / 8 ILE A 354
GLU A 369
GLN A 352
LEU A 370
None
0.85A 4mj8A-3s95A:
undetectable
4mj8A-3s95A:
19.42
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXO_A_DB8A601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LEU A 345
LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
ASP A 478
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 ( 4.2A)
0.80A 4mxoA-3s95A:
26.9
4mxoA-3s95A:
34.83
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXO_B_DB8B601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LEU A 345
LYS A 368
GLU A 384
THR A 413
TYR A 415
GLY A 419
LEU A 467
ASP A 478
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.2A)
0.82A 4mxoB-3s95A:
27.0
4mxoB-3s95A:
34.83
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4MXX_A_DB8A601_1
(PROTO-ONCOGENE
TYROSINE-PROTEIN
KINASE SRC)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.75A 4mxxA-3s95A:
20.3
4mxxA-3s95A:
34.53
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4O0S_A_ADNA500_1
(AURORA KINASE A)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 11 LEU A 345
GLY A 346
LYS A 368
LEU A 397
THR A 420
ASN A 465
LEU A 467
STU  A   1 (-3.8A)
STU  A   1 (-3.4A)
STU  A   1 (-3.1A)
STU  A   1 (-4.6A)
STU  A   1 (-4.6A)
STU  A   1 (-4.5A)
STU  A   1 (-4.6A)
0.85A 4o0sA-3s95A:
26.9
4o0sA-3s95A:
27.52
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4OTW_A_DB8A1101_1
(RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
LYS A 368
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.79A 4otwA-3s95A:
23.6
4otwA-3s95A:
25.22
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4OTW_A_DB8A1101_1
(RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-3)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
ASP A 478
STU  A   1 (-3.8A)
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
STU  A   1 ( 4.2A)
0.77A 4otwA-3s95A:
23.6
4otwA-3s95A:
25.22
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4QB9_D_PARD500_1
(ENHANCED
INTRACELLULAR
SURVIVAL PROTEIN)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
4 / 8 PHE A 597
SER A 534
GLU A 384
ASP A 478
None
None
STU  A   1 (-3.7A)
STU  A   1 ( 4.2A)
1.31A 4qb9D-3s95A:
undetectable
4qb9D-3s95A:
22.62
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4QRC_A_0LIA802_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 4)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 12 GLU A 384
MET A 388
LEU A 451
ARG A 459
ALA A 477
STU  A   1 (-3.7A)
None
None
None
STU  A   1 ( 4.1A)
1.02A 4qrcA-3s95A:
26.1
4qrcA-3s95A:
29.64
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4RTB_A_SAMA501_1
(HYDG PROTEIN)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 GLU A 630
ARG A 633
GLN A 623
None
0.88A 4rtbA-3s95A:
undetectable
4rtbA-3s95A:
20.74
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4UXQ_A_0LIA1752_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 4)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 12 LEU A 345
LEU A 451
HIS A 458
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
None
None
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.26A 4uxqA-3s95A:
25.9
4uxqA-3s95A:
30.17
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V04_A_0LIA1772_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 8 LYS A 368
MET A 388
TYR A 415
ARG A 459
LEU A 467
STU  A   1 (-3.1A)
None
STU  A   1 (-4.7A)
None
STU  A   1 (-4.6A)
1.24A 4v04A-3s95A:
25.4
4v04A-3s95A:
30.50
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4V04_B_0LIB1771_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1
(FMS-RELATED
TYROSINE KINASE 2,
PFEIFFER SYNDROME),
ISOFORM CRA_B)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 10 LEU A 345
LYS A 368
MET A 388
TYR A 415
ARG A 459
LEU A 467
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
None
STU  A   1 (-4.7A)
None
STU  A   1 (-4.6A)
1.17A 4v04B-3s95A:
26.0
4v04B-3s95A:
30.50
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4WKQ_A_IREA1101_1
(EPIDERMAL GROWTH
FACTOR RECEPTOR)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LEU A 345
LYS A 368
GLU A 384
MET A 388
THR A 413
GLY A 419
LEU A 467
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.97A 4wkqA-3s95A:
26.8
4wkqA-3s95A:
28.12
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4XLI_A_1N1A601_1
(NON-SPECIFIC
PROTEIN-TYROSINE
KINASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
9 / 12 LEU A 345
LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.76A 4xliA-3s95A:
27.5
4xliA-3s95A:
31.45
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4XLI_B_1N1B600_1
(NON-SPECIFIC
PROTEIN-TYROSINE
KINASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
9 / 12 LEU A 345
LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.67A 4xliB-3s95A:
27.2
4xliB-3s95A:
31.45
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XV2_B_P06B801_1
(SERINE/THREONINE-PRO
TEIN KINASE B-RAF)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 12 LYS A 368
LEU A 397
THR A 413
ASP A 478
PHE A 479
STU  A   1 (-3.1A)
STU  A   1 (-4.6A)
STU  A   1 (-3.9A)
STU  A   1 ( 4.2A)
None
0.84A 4xv2B-3s95A:
25.1
4xv2B-3s95A:
29.62
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5BVW_A_1N1A1009_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LEU A 345
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.85A 5bvwA-3s95A:
24.5
5bvwA-3s95A:
28.42
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5BVW_A_1N1A1009_1
(EPITHELIAL DISCOIDIN
DOMAIN-CONTAINING
RECEPTOR 1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
8 / 12 LEU A 345
LYS A 368
GLU A 384
THR A 413
TYR A 415
GLY A 419
LEU A 467
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.1A)
0.68A 5bvwA-3s95A:
24.5
5bvwA-3s95A:
28.42
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5DV4_A_NMYA601_1
(CCR4-NOT
TRANSCRIPTION
COMPLEX SUBUNIT
6-LIKE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 12 LEU A 391
ASN A 462
ASP A 531
ILE A 457
HIS A 452
None
1.21A 5dv4A-3s95A:
undetectable
5dv4A-3s95A:
22.06
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5F9Z_B_HFGB703_0
(AMINOACYL-TRNA
SYNTHETASE)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 12 LEU A 600
PHE A 535
VAL A 532
PRO A 595
GLY A 627
None
None
None
GOL  A   6 ( 4.6A)
None
1.33A 5f9zB-3s95A:
undetectable
5f9zB-3s95A:
20.97
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5HI2_A_BAXA801_1
(SERINE/THREONINE-PRO
TEIN KINASE B-RAF)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 12 LYS A 368
GLU A 384
LEU A 397
THR A 413
LEU A 451
HIS A 458
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-4.6A)
STU  A   1 (-3.9A)
None
None
0.62A 5hi2A-3s95A:
25.7
5hi2A-3s95A:
29.47
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5I9X_A_DB8A1001_1
(EPHRIN TYPE-A
RECEPTOR 2)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 12 LYS A 368
GLU A 384
THR A 413
TYR A 415
GLY A 419
LEU A 467
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.72A 5i9xA-3s95A:
26.4
5i9xA-3s95A:
29.81
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5I9Y_A_1N1A1001_1
(EPHRIN TYPE-A
RECEPTOR 2)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
7 / 12 LYS A 368
GLU A 384
MET A 388
THR A 413
TYR A 415
GLY A 419
LEU A 467
STU  A   1 (-3.1A)
STU  A   1 (-3.7A)
None
STU  A   1 (-3.9A)
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 (-4.6A)
0.75A 5i9yA-3s95A:
19.1
5i9yA-3s95A:
29.81
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5IEN_B_VDYB201_1
(CDL2.2)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
5 / 10 PRO A 433
VAL A 468
ILE A 542
LEU A 421
LEU A 607
None
1.13A 5ienB-3s95A:
undetectable
5ienB-3s95A:
20.97
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5ZV2_A_LEVA801_1
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
6 / 12 LEU A 345
GLU A 384
MET A 388
TYR A 415
GLY A 419
ALA A 477
STU  A   1 (-3.8A)
STU  A   1 (-3.7A)
None
STU  A   1 (-4.7A)
STU  A   1 (-3.6A)
STU  A   1 ( 4.1A)
0.80A 5zv2A-3s95A:
25.0
5zv2A-3s95A:
14.33
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5ZV2_A_LEVA801_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 LYS A 368
LEU A 467
ASP A 478
STU  A   1 (-3.1A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.2A)
0.76A 5zv2A-3s95A:
25.0
5zv2A-3s95A:
14.33
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
5ZV2_B_LEVB801_2
(FIBROBLAST GROWTH
FACTOR RECEPTOR 1)
3s95 LIM DOMAIN KINASE 1
(Homo
sapiens)
3 / 3 TYR A 415
LEU A 467
ASP A 478
STU  A   1 (-4.7A)
STU  A   1 (-4.6A)
STU  A   1 ( 4.2A)
0.64A 5zv2B-3s95A:
25.1
5zv2B-3s95A:
14.33