SIMILAR PATTERN OF AMINO ACIDS MAPPED TO '4j5x'

List of Similar Pattern of Amino Acids

Hit pattern: 3D amino acid arrangements similar to known drug binding site

Query pattern: Residues from known binding site for annotated drug that match the hit pattern


(Click on the DrReposER ID to view details on interfaces and similar patterns of amino acids)
(Click on the view link on the last column to view superposed patterns of amino acids)
Filter list by:
DrReposER ID / Desc. Hit
PDBID
Hit
Macromolecule
Res.
Matches
Interface HETATM RMSD Dali
Z-score
Seq.
Identity (%)
View Dock
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1ERR_A_RALA600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 276
TRP D 305
ARG D 316
ILE D 428
None
1.05A 1errA-4j5xD:
22.2
1errA-4j5xD:
29.51
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1ERR_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 276
TRP D 305
ARG D 316
ILE D 428
None
1.01A 1errB-4j5xD:
22.7
1errB-4j5xD:
29.51
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
1ERR_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
ILE D 428
None
0.91A 1errB-4j5xD:
22.7
1errB-4j5xD:
29.51
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FBY_A_9CRA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
CYH D 269
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
HIS D 435
None
0.61A 1fbyA-4j5xD:
32.2
1fbyA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FBY_B_9CRB1500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
CYH D 269
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
HIS D 435
None
0.59A 1fbyB-4j5xD:
31.5
1fbyB-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM6_A_9CRA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 271
ALA D 272
GLN D 275
TRP D 305
ARG D 316
LEU D 455
None
1.42A 1fm6A-4j5xD:
32.3
1fm6A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM6_A_9CRA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.59A 1fm6A-4j5xD:
32.3
1fm6A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM6_U_9CRU502_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 12 ALA D 271
ALA D 272
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
ILE D 345
CYH D 432
HIS D 435
LEU D 436
None
0.60A 1fm6U-4j5xD:
32.4
1fm6U-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM6_U_9CRU502_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 PHE D 313
ARG D 316
ILE D 345
CYH D 432
HIS D 435
LEU D 433
None
1.34A 1fm6U-4j5xD:
32.4
1fm6U-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM6_U_9CRU502_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 TRP D 305
VAL D 342
ILE D 345
CYH D 432
HIS D 435
LEU D 436
None
1.12A 1fm6U-4j5xD:
32.4
1fm6U-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM9_A_9CRA201_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
7 / 12 ALA D 271
ALA D 272
TRP D 305
LEU D 309
ARG D 316
ALA D 327
LEU D 455
None
1.35A 1fm9A-4j5xD:
33.0
1fm9A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM9_A_9CRA201_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.55A 1fm9A-4j5xD:
33.0
1fm9A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1FM9_A_9CRA201_2
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
3 / 3 GLN D 275
ILE D 345
HIS D 435
None
0.42A 1fm9A-4j5xD:
33.0
1fm9A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1G5Y_C_9CRC502_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 10 LEU D 309
SER D 312
PHE D 313
ARG D 316
LEU D 326
ALA D 327
None
0.67A 1g5yC-4j5xD:
25.4
1g5yC-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1K74_A_9CRA463_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
7 / 12 ALA D 271
ALA D 272
TRP D 305
LEU D 309
ARG D 316
ALA D 327
LEU D 455
None
1.39A 1k74A-4j5xD:
32.8
1k74A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1K74_A_9CRA463_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.58A 1k74A-4j5xD:
32.8
1k74A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1K74_A_9CRA463_2
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
3 / 3 GLN D 275
ILE D 345
HIS D 435
None
0.39A 1k74A-4j5xD:
32.8
1k74A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1QKN_A_RALA600_1
(ESTROGEN RECEPTOR
BETA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
LEU D 309
ARG D 316
ILE D 345
ILE D 428
GLY D 429
None
1.01A 1qknA-4j5xD:
23.1
1qknA-4j5xD:
30.66
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XDK_A_9CRA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 12 ILE D 268
ALA D 271
GLN D 275
TRP D 305
ASN D 306
PHE D 313
ARG D 316
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.71A 1xdkA-4j5xD:
34.1
1xdkA-4j5xD:
99.15
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XDK_A_9CRA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 12 ILE D 268
ALA D 271
GLN D 275
TRP D 305
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.60A 1xdkA-4j5xD:
34.1
1xdkA-4j5xD:
99.15
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XDK_E_9CRE1500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.58A 1xdkE-4j5xD:
34.1
1xdkE-4j5xD:
99.15
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XDK_E_9CRE1500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ILE D 268
ALA D 271
GLN D 275
PHE D 313
VAL D 342
CYH D 432
None
1.44A 1xdkE-4j5xD:
34.1
1xdkE-4j5xD:
99.15
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XIU_A_9CRA201_1
(RXR-LIKE PROTEIN)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
CYH D 269
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.55A 1xiuA-4j5xD:
30.5
1xiuA-4j5xD:
77.82
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XIU_B_9CRB202_1
(RXR-LIKE PROTEIN)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
LEU D 309
PHE D 313
ARG D 316
ALA D 327
VAL D 342
CYH D 432
HIS D 435
LEU D 436
None
0.48A 1xiuB-4j5xD:
34.3
1xiuB-4j5xD:
77.82
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XIU_B_9CRB202_1
(RXR-LIKE PROTEIN)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ILE D 268
ALA D 271
GLN D 275
PHE D 313
VAL D 342
HIS D 435
None
1.47A 1xiuB-4j5xD:
34.3
1xiuB-4j5xD:
77.82
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XLS_A_9CRA801_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.48A 1xlsA-4j5xD:
33.6
1xlsA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XLS_B_9CRB802_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.48A 1xlsB-4j5xD:
33.5
1xlsB-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XLS_C_9CRC803_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.48A 1xlsC-4j5xD:
33.5
1xlsC-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
1XLS_D_9CRD804_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.48A 1xlsD-4j5xD:
33.6
1xlsD-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ACL_A_REAA502_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 12 ALA D 271
ALA D 272
GLN D 275
ASN D 306
LEU D 309
PHE D 313
ARG D 316
ALA D 327
ILE D 345
CYH D 432
None
0.76A 2aclA-4j5xD:
28.4
2aclE-4j5xD:
28.3
2aclA-4j5xD:
100.00
2aclE-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ACL_A_REAA502_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 12 ALA D 271
ALA D 272
GLN D 275
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
ILE D 345
CYH D 432
None
0.72A 2aclA-4j5xD:
28.4
2aclE-4j5xD:
28.3
2aclA-4j5xD:
100.00
2aclE-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ACL_C_REAC503_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 10 ILE D 268
ALA D 271
ALA D 272
GLN D 275
ASN D 306
PHE D 313
ARG D 316
ALA D 327
ILE D 345
CYH D 432
None
0.77A 2aclC-4j5xD:
28.5
2aclC-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ACL_E_REAE504_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 11 ILE D 268
ALA D 271
ALA D 272
GLN D 275
ASN D 306
LEU D 309
PHE D 313
ARG D 316
ALA D 327
ILE D 345
CYH D 432
None
0.80A 2aclE-4j5xD:
28.3
2aclE-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
2ACL_G_REAG501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
ASN D 306
LEU D 309
ILE D 310
PHE D 313
ARG D 316
LEU D 326
ALA D 327
CYH D 432
None
0.76A 2aclG-4j5xD:
27.7
2aclG-4j5xD:
100.00
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2JFA_A_RALA600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
LEU D 276
TRP D 305
LEU D 309
ARG D 316
ILE D 345
None
0.96A 2jfaA-4j5xD:
21.6
2jfaA-4j5xD:
25.26
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2JFA_A_RALA600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
LEU D 276
TRP D 305
LEU D 309
ARG D 316
ILE D 428
None
1.08A 2jfaA-4j5xD:
21.6
2jfaA-4j5xD:
25.26
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2JFA_A_RALA600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
ILE D 345
LEU D 436
None
0.90A 2jfaA-4j5xD:
21.6
2jfaA-4j5xD:
25.26
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2JFA_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
LEU D 276
TRP D 305
LEU D 309
ARG D 316
GLY D 429
None
0.94A 2jfaB-4j5xD:
21.2
2jfaB-4j5xD:
25.26
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2JFA_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
LEU D 436
None
0.80A 2jfaB-4j5xD:
21.2
2jfaB-4j5xD:
25.26
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2NV4_A_ACTA148_0
(UPF0066 PROTEIN
AF_0241)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
3 / 3 VAL D 242
GLU D 239
GLU D 243
None
0.73A 2nv4A-4j5xD:
undetectable
2nv4A-4j5xD:
21.96
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2QXS_A_RALA600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
LEU D 276
TRP D 305
LEU D 309
ARG D 316
ILE D 345
None
1.01A 2qxsA-4j5xD:
23.5
2qxsA-4j5xD:
29.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2QXS_A_RALA600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
LEU D 276
TRP D 305
LEU D 309
ARG D 316
ILE D 428
None
1.08A 2qxsA-4j5xD:
23.5
2qxsA-4j5xD:
29.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2QXS_A_RALA600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
ILE D 345
LEU D 436
None
0.90A 2qxsA-4j5xD:
23.5
2qxsA-4j5xD:
29.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2QXS_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 276
TRP D 305
ARG D 316
ILE D 345
None
0.90A 2qxsB-4j5xD:
23.1
2qxsB-4j5xD:
29.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2QXS_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 276
TRP D 305
ARG D 316
ILE D 428
None
1.10A 2qxsB-4j5xD:
23.1
2qxsB-4j5xD:
29.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2QXS_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
ILE D 345
LEU D 436
None
0.93A 2qxsB-4j5xD:
23.1
2qxsB-4j5xD:
29.72
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
2QXS_B_RALB600_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
ILE D 428
None
0.92A 2qxsB-4j5xD:
23.1
2qxsB-4j5xD:
29.72
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3DZU_A_9CRA7223_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
GLN D 275
ASN D 306
ILE D 310
PHE D 313
ARG D 316
LEU D 326
VAL D 342
CYH D 432
HIS D 435
LEU D 436
None
0.68A 3dzuA-4j5xD:
31.7
3dzuA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3DZY_A_9CRA463_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
8 / 12 GLN D 275
ASN D 306
SER D 312
ARG D 316
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.91A 3dzyA-4j5xD:
30.1
3dzyA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3DZY_A_9CRA463_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 12 ILE D 268
ALA D 271
GLN D 275
ASN D 306
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.71A 3dzyA-4j5xD:
30.1
3dzyA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3E00_A_9CRA7223_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
ASN D 306
PHE D 313
ALA D 327
VAL D 342
ILE D 345
CYH D 432
None
0.67A 3e00A-4j5xD:
32.2
3e00A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3E00_A_9CRA7223_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
PHE D 313
ARG D 316
ALA D 327
VAL D 342
ILE D 345
CYH D 432
None
0.58A 3e00A-4j5xD:
32.2
3e00A-4j5xD:
100.00
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3ERD_A_DESA600_1
(ESTROGEN RECEPTOR
ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 309
ARG D 316
HIS D 435
LEU D 436
None
1.01A 3erdA-4j5xD:
24.3
3erdA-4j5xD:
28.32
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3ERD_B_DESB800_1
(ESTROGEN RECEPTOR
ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 10 ALA D 272
LEU D 309
ARG D 316
HIS D 435
LEU D 436
None
0.99A 3erdB-4j5xD:
25.0
3erdB-4j5xD:
28.32
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3FAL_A_REAA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 10 ILE D 268
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
ALA D 327
VAL D 342
ILE D 345
CYH D 432
None
0.57A 3falA-4j5xD:
27.8
3falA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3FAL_A_REAA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
7 / 10 ILE D 268
ALA D 271
GLN D 275
PHE D 313
VAL D 342
ILE D 345
CYH D 432
None
1.45A 3falA-4j5xD:
27.8
3falA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3FAL_C_REAC501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 10 ILE D 268
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
LEU D 326
ALA D 327
ILE D 345
CYH D 432
None
0.64A 3falC-4j5xD:
28.0
3falC-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3FC6_A_REAA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 11 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
PHE D 313
ARG D 316
LEU D 326
ALA D 327
ILE D 345
CYH D 432
None
0.63A 3fc6A-4j5xD:
28.7
3fc6A-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3FC6_C_REAC501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 VAL D 265
CYH D 269
ALA D 271
ALA D 272
GLN D 275
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
None
0.64A 3fc6C-4j5xD:
29.0
3fc6C-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3H0A_A_9RAA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
9 / 12 ALA D 271
ALA D 272
GLN D 275
LEU D 309
ARG D 316
LEU D 326
VAL D 342
ILE D 345
CYH D 432
None
0.87A 3h0aA-4j5xD:
30.9
3h0aA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3H0A_A_9RAA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 12 ALA D 271
ALA D 272
GLN D 275
TRP D 305
LEU D 309
ARG D 316
LEU D 326
VAL D 342
ILE D 345
LEU D 436
None
0.67A 3h0aA-4j5xD:
30.9
3h0aA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3H0A_A_9RAA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
9 / 12 ALA D 271
GLN D 275
LEU D 309
ARG D 316
LEU D 326
ALA D 327
VAL D 342
ILE D 345
CYH D 432
None
0.99A 3h0aA-4j5xD:
30.9
3h0aA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3H0A_A_9RAA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
7 / 12 ALA D 271
GLN D 275
TRP D 305
ARG D 316
LEU D 326
ALA D 327
ILE D 428
None
1.43A 3h0aA-4j5xD:
30.9
3h0aA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3H0A_A_9RAA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 12 ALA D 271
GLN D 275
TRP D 305
LEU D 309
ARG D 316
LEU D 326
ALA D 327
VAL D 342
ILE D 345
LEU D 436
None
0.80A 3h0aA-4j5xD:
30.9
3h0aA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3H0A_A_9RAA500_2
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
3 / 3 ILE D 268
PHE D 313
HIS D 435
None
0.61A 3h0aA-4j5xD:
30.9
3h0aA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OAP_A_9CRA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 GLN D 275
PHE D 313
ARG D 316
ILE D 345
CYH D 432
LEU D 433
None
1.46A 3oapA-4j5xD:
34.6
3oapA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3OAP_A_9CRA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
ILE D 345
CYH D 432
LEU D 436
None
0.56A 3oapA-4j5xD:
34.6
3oapA-4j5xD:
100.00
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3OLS_B_ESTB600_1
(ESTROGEN RECEPTOR
BETA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 309
ARG D 316
ILE D 345
LEU D 436
None
1.03A 3olsB-4j5xD:
24.4
3olsB-4j5xD:
28.62
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3Q95_A_ESLA700_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 309
ARG D 316
ILE D 345
LEU D 436
None
0.97A 3q95A-4j5xD:
24.5
3q95A-4j5xD:
28.91
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3Q95_A_ESLA700_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 309
ARG D 316
ILE D 428
GLY D 429
None
0.96A 3q95A-4j5xD:
24.5
3q95A-4j5xD:
28.91
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3Q95_B_ESLB700_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 309
ARG D 316
ILE D 345
LEU D 436
None
0.95A 3q95B-4j5xD:
23.9
3q95B-4j5xD:
28.91
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
3Q95_B_ESLB700_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
LEU D 309
ARG D 316
ILE D 428
GLY D 429
None
0.98A 3q95B-4j5xD:
23.9
3q95B-4j5xD:
28.91
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
3UVV_B_9CRB501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
LEU D 309
PHE D 313
ARG D 316
ALA D 327
VAL D 342
ILE D 345
CYH D 432
LEU D 436
None
0.48A 3uvvB-4j5xD:
35.4
3uvvB-4j5xD:
95.56
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4J24_D_ESTD600_1
(ESTROGEN RECEPTOR
BETA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
ARG D 316
ILE D 345
HIS D 435
LEU D 436
None
1.11A 4j24D-4j5xD:
24.1
4j24D-4j5xD:
28.62
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4K6I_A_9RAA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
LEU D 309
ILE D 310
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 349
None
0.55A 4k6iA-4j5xD:
34.4
4k6iA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4K6I_A_9RAA500_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
9 / 12 ILE D 268
ALA D 271
GLN D 275
ILE D 310
PHE D 313
ARG D 316
LEU D 326
ALA D 327
CYH D 432
None
0.84A 4k6iA-4j5xD:
34.4
4k6iA-4j5xD:
100.00
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4L1A_A_AB1A101_1
(MDR769 HIV-1
PROTEASE)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 11 GLY D 341
ALA D 340
ILE D 324
THR D 266
THR D 445
None
1.08A 4l1aA-4j5xD:
undetectable
4l1aA-4j5xD:
16.28
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4NQA_A_9CRA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 11 ILE D 268
ALA D 272
GLN D 275
PHE D 313
ARG D 316
ALA D 327
None
0.73A 4nqaA-4j5xD:
33.3
4nqaA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4NQA_A_9CRA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
10 / 11 ILE D 268
ALA D 272
GLN D 275
PHE D 313
LEU D 326
ALA D 327
VAL D 342
CYH D 432
HIS D 435
LEU D 436
None
0.74A 4nqaA-4j5xD:
33.3
4nqaA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4NQA_H_9CRH501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
9 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
LEU D 326
ALA D 327
LEU D 436
None
0.58A 4nqaH-4j5xD:
33.2
4nqaH-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4NQA_H_9CRH501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
7 / 12 ILE D 268
ALA D 271
ALA D 272
ILE D 345
CYH D 432
HIS D 435
LEU D 436
None
0.65A 4nqaH-4j5xD:
33.2
4nqaH-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
4NQA_H_9CRH501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
9 / 12 ILE D 268
ALA D 271
ALA D 272
PHE D 313
ARG D 316
ALA D 327
CYH D 432
HIS D 435
LEU D 436
None
0.66A 4nqaH-4j5xD:
33.2
4nqaH-4j5xD:
100.00
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XI3_B_29SB601_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
LEU D 276
TRP D 305
ARG D 316
ILE D 428
GLY D 429
None
1.12A 4xi3B-4j5xD:
23.0
4xi3B-4j5xD:
29.14
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XI3_B_29SB601_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
6 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
ILE D 428
GLY D 429
None
0.98A 4xi3B-4j5xD:
23.0
4xi3B-4j5xD:
29.14
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XI3_B_29SB601_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ASP D 273
TRP D 305
LEU D 309
ARG D 316
LEU D 436
None
0.99A 4xi3B-4j5xD:
23.0
4xi3B-4j5xD:
29.14
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XI3_C_29SC601_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
GLY D 429
None
0.83A 4xi3C-4j5xD:
22.8
4xi3C-4j5xD:
29.14
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
4XI3_D_29SD601_1
(ESTROGEN RECEPTOR)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
5 / 12 ALA D 272
TRP D 305
LEU D 309
ARG D 316
LEU D 436
None
0.91A 4xi3D-4j5xD:
22.7
4xi3D-4j5xD:
29.14
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5JI0_A_9CRA501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
11 / 11 ILE D 268
GLN D 275
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.52A 5ji0A-4j5xD:
32.4
5ji0A-4j5xD:
99.58
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5UAN_A_9CRA503_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.74A 5uanA-4j5xD:
32.3
5uanA-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5Z12_B_9CRB501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
TRP D 305
LEU D 309
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.51A 5z12B-4j5xD:
34.2
5z12B-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5Z12_B_9CRB501_2
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
3 / 3 GLN D 275
ILE D 345
HIS D 435
None
0.50A 5z12B-4j5xD:
34.2
5z12B-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
5Z12_C_9CRC501_1
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
PHE D 313
ARG D 316
LEU D 326
ALA D 327
VAL D 342
CYH D 432
LEU D 436
None
0.60A 5z12C-4j5xD:
32.0
5z12C-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A5Y_D_9CRD501_0
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
7 / 12 ALA D 271
ALA D 272
GLN D 275
TRP D 305
ARG D 316
ALA D 327
LEU D 455
None
1.28A 6a5yD-4j5xD:
33.9
6a5yD-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A5Y_D_9CRD501_0
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
TRP D 305
PHE D 313
ARG D 316
LEU D 326
ALA D 327
ILE D 345
CYH D 432
LEU D 436
None
0.57A 6a5yD-4j5xD:
33.9
6a5yD-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A5Z_D_9CRD501_0
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
ILE D 310
PHE D 313
ARG D 316
LEU D 326
ALA D 327
ILE D 345
CYH D 432
LEU D 436
None
0.52A 6a5zD-4j5xD:
33.9
6a5zD-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A5Z_L_9CRL501_0
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
PHE D 313
ARG D 316
LEU D 326
ALA D 327
ILE D 345
CYH D 432
HIS D 435
LEU D 436
None
0.56A 6a5zL-4j5xD:
33.3
6a5zL-4j5xD:
100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A60_D_9CRD501_0
(RETINOIC ACID
RECEPTOR RXR-ALPHA)
4j5x RETINOIC ACID
RECEPTOR RXR-ALPHA,
NUCLEAR RECEPTOR
COACTIVATOR 1

(Homo
sapiens)
12 / 12 ILE D 268
ALA D 271
ALA D 272
GLN D 275
LEU D 309
PHE D 313
ARG D 316
ALA D 327
ILE D 345
CYH D 432
HIS D 435
LEU D 436
None
0.48A 6a60D-4j5xD:
33.8
6a60D-4j5xD:
100.00